BAYESPHARMA · INNOVATORLEAD OPTIMIZATION PROGRAMME v2
← Discovery Programme
Measured SAR · Design–Make–Test–Learn

Lead Optimization Programme

Start from a human-confirmed experimental hit, organize a persistent chemical series, learn from approved measured assays, register explicit analogue hypotheses, select only evidence-ready compounds for Make/Test, and keep every cycle linked back to the same programme.

Measured data is primary truthNo invented potency gainsRDKit identity + similarityADMET + synthesis gateHuman progression decisions
01 Discover
02 Hit Review
03 CRO
04 Measured Results
05 Confirm Hit
06 Lead Optimization
07 Lead Progression

Lead series

A series can only be seeded from an experimentally confirmed hit with approved measured assay evidence.

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